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Molecular Determinants of hERG Channel Block by Terfenadine and Cisapride

Block of cardiac hERG K(+) channels by the antihistamine terfenadine and the prokinetic agent cisapride is associated with prolonged ventricular repolarization and an increased risk of ventricular arrhythmia. Here, we used a site-directed mutagenesis approach to determine the molecular determinants...

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Bibliografske podrobnosti
Main Authors: Kamiya, Kaichiro, Niwa, Ryoko, Morishima, Mikio, Honjo, Haruo, Sanguinetti, Michael C.
Format: Artigo
Jezik:Inglês
Izdano: 2008
Teme:
Online dostop:https://ncbi.nlm.nih.gov/pmc/articles/PMC2845965/
https://ncbi.nlm.nih.gov/pubmed/18987434
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