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C6 –C8 Bridged Epothilones: Consequences of Installing a Conformational Lock at the Edge of the Macrocycle

A series of conformationally restrained epothilone analogs with a short bridge between the methyl groups at C6 and C8 was designed to mimic the binding pose assigned to our recently reported EpoA-microtubule binding model. A versatile synthetic route to these bridged epothilone analogs has been succ...

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Detalhes bibliográficos
Main Authors: Zhan, Weiqiang, Jiang, Yi, Banerjee, Abhijit, Brodie, Peggy J., Bane, Susan, Kingston, David G. I., Liotta, Dennis C., Snyder, James P.
Formato: Artigo
Idioma:Inglês
Publicado em: 2011
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC3248799/
https://ncbi.nlm.nih.gov/pubmed/22127984
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1002/chem.201102630
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