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Design, synthesis and biological evaluation of bridged epothilone D analogues†

Six epothilone D analogues with a bridge between the C4-methyl and the C12-methyl carbons were prepared in an attempt to constrain epothilone D to its proposed tubulin-binding conformation. Ring-closing metathesis (RCM) was employed as the key step to build the C4-C26 bridge. In antiproliferative as...

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Detalhes bibliográficos
Main Authors: Chen, Qiao-Hong, Ganesh, Thota, Brodie, Peggy, Slebodnick, Carla, Jiang, Yi, Banerjee, Abhijit, Bane, Susan, Snyder, James P., Kingston, David G. I.
Formato: Artigo
Idioma:Inglês
Publicado em: 2008
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC2790820/
https://ncbi.nlm.nih.gov/pubmed/19039362
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1039/b814823f
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