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Design and Synthesis of C6–C8 Bridged Epothilone A

[Image: see text] A conformationally restrained epothilone A analogue (3) with a short bridge between methyl groups at C6 and C8 was designed and synthesized. Preliminary biological evaluation indicates 3 to be only weakly active (IC(50) = 8.5 µM) against the A2780 human ovarian cancer cell line.

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Detalhes bibliográficos
Main Authors: Zhan, Weiqiang, Jiang, Yi, Brodie, Peggy J., Kingston, David G. I., Liotta, Dennis C., Snyder, James P.
Formato: Artigo
Idioma:Inglês
Publicado em: 2008
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC3249659/
https://ncbi.nlm.nih.gov/pubmed/18355076
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/ol800422q
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