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Mechanism-Based Inactivation by Aromatization of the Transaminase BioA Involved in Biotin Biosynthesis in Mycobaterium tuberculosis

BioA catalyzes the second step of biotin biosynthesis and this enzyme represents a potential target to develop new antitubercular agents. Herein we report the design, synthesis, and biochemical characterization of a mechanism-based inhibitor (1) featuring a 3,6-dihydropyrid-2-one heterocycle that co...

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Main Authors: Shi, Ce, Geders, Todd W., Park, Sae Woong, Wilson, Daniel J., Boshoff, Helena I., Orisadipe, Abayomi, Barry, Clifton E., Schnappinger, Dirk, Finzel, Barry C., Aldrich, Courtney C.
格式: Artigo
語言:Inglês
出版: 2011
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在線閱讀:https://ncbi.nlm.nih.gov/pmc/articles/PMC3222238/
https://ncbi.nlm.nih.gov/pubmed/21988601
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/ja204036t
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