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Selection of Cyclic-Peptide Inhibitors Targeting Aurora Kinase A: Problems and Solutions

The critical role of Aurora kinase in cell cycle progression and its deregulation in cancer has garnered significant interest. As such, numerous Aurora targeted inhibitors have been developed to date, almost all of which target the ATP cleft at the active site. These current inhibitors display polyp...

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Bibliographic Details
Main Authors: Shomin, Carolyn D., Restituyo, Elizabeth, Cox, Kurt J., Ghosh, Indraneel
Format: Artigo
Language:Inglês
Published: 2011
Subjects:
Online Access:https://ncbi.nlm.nih.gov/pmc/articles/PMC3206593/
https://ncbi.nlm.nih.gov/pubmed/22004849
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.bmc.2011.09.049
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