A carregar...

Staurosporine Tethered Peptide Ligands that Target cAMP-dependent Protein Kinase (PKA): Optimization and Selectivity Profiling

We have recently developed a fragment based selection strategy for targeting kinases, where a small molecule warhead can be non-covalently tethered to a phage-displayed library of peptides. This approach was applied to the conversion of the promiscuous kinase inhibitor, staurosporine, into a potent...

ver descrição completa

Na minha lista:
Detalhes bibliográficos
Main Authors: Shomin, Carolyn D., Meyer, Scott C., Ghosh, Indraneel
Formato: Artigo
Idioma:Inglês
Publicado em: 2009
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC2749490/
https://ncbi.nlm.nih.gov/pubmed/19674907
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.bmc.2009.07.056
Tags: Adicionar Tag
Sem tags, seja o primeiro a adicionar uma tag!