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Molecular Determinants for Activation of Human Ether-à-go-go-related Gene 1 Potassium Channels by 3-Nitro-N-(4-phenoxyphenyl) Benzamide

Human ether-à-go-go-related gene 1 (hERG1) channels mediate repolarization of cardiac action potentials. Inherited long QT syndrome (LQTS) caused by loss-of-function mutations, or unintended blockade of hERG1 channels by many drugs, can lead to severe arrhythmia and sudden death. Drugs that activate...

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Bibliographic Details
Main Authors: Garg, Vivek, Stary-Weinzinger, Anna, Sachse, Frank, Sanguinetti, Michael C.
Format: Artigo
Language:Inglês
Published: The American Society for Pharmacology and Experimental Therapeutics 2011
Subjects:
Online Access:https://ncbi.nlm.nih.gov/pmc/articles/PMC3187531/
https://ncbi.nlm.nih.gov/pubmed/21743002
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1124/mol.111.073809
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