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Structural study of phenyl boronic acid derivatives as AmpC β-lactamase inhibitors

A small set of boronic acids acting as low nanomolar inhibitors of AmpC β-lactamase were designed and synthesized in the effort to improve affinity, pharmacokinetic properties, and to provide a valid lead compound. X-ray crystallography revealed the binary complex of the best inhibitor bound to the...

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Autori principali: Tondi, Donatella, Calò, Samuele, Shoichet, Brian K., Costi, Maria Paola
Natura: Artigo
Lingua:Inglês
Pubblicazione: 2010
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC3177945/
https://ncbi.nlm.nih.gov/pubmed/20452208
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.bmcl.2010.04.007
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