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The 8-Aminoquinoline Analogue Sitamaquine Causes Oxidative Stress in Leishmania donovani Promastigotes by Targeting Succinate Dehydrogenase

The 8-aminoquinoline analogue sitamaquine (SQ) is an oral antileishmanial drug currently undergoing phase 2b clinical trials for the treatment of visceral leishmaniasis. In the present study, we investigated the mechanism of action of this drug in Leishmania donovani promastigotes. SQ causes a dose-...

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Autori principali: Carvalho, Luis, Luque-Ortega, Juan Román, López-Martín, Carmen, Castanys, Santiago, Rivas, Luis, Gamarro, Francisco
Natura: Artigo
Lingua:Inglês
Pubblicazione: American Society for Microbiology 2011
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC3165367/
https://ncbi.nlm.nih.gov/pubmed/21670183
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1128/AAC.00520-11
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