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The 8-Aminoquinoline Analogue Sitamaquine Causes Oxidative Stress in Leishmania donovani Promastigotes by Targeting Succinate Dehydrogenase

The 8-aminoquinoline analogue sitamaquine (SQ) is an oral antileishmanial drug currently undergoing phase 2b clinical trials for the treatment of visceral leishmaniasis. In the present study, we investigated the mechanism of action of this drug in Leishmania donovani promastigotes. SQ causes a dose-...

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Autors principals: Carvalho, Luis, Luque-Ortega, Juan Román, López-Martín, Carmen, Castanys, Santiago, Rivas, Luis, Gamarro, Francisco
Format: Artigo
Idioma:Inglês
Publicat: American Society for Microbiology 2011
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Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC3165367/
https://ncbi.nlm.nih.gov/pubmed/21670183
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1128/AAC.00520-11
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