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Preparation of a Series of 5-Methyl-3-(substituted)-[1,2,4]triazines

Procedures for the synthesis of thirty-six 5-methyl-3-(substituted)-[1,2,4]triazines have been described. These compounds were evaluated for antagonism at metabotropic glutamate receptor subtype 5. Two compounds, 5b and 3c, were determined to be low micromolar inhibitors of mGluR5.

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Autors principals: Gichinga, Moses G., Olson, Jeremy P., Butala, Elizabeth, Gilmour, Brian P., Navarro, Hernán H., Carroll, F. Ivy
Format: Artigo
Idioma:Inglês
Publicat: 2011
Matèries:
Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC3138555/
https://ncbi.nlm.nih.gov/pubmed/21779134
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.tetlet.2011.04.075
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