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In Vivo and In Vitro Characterization of a First-in-Class Novel Azole Analog That Targets Pregnane X Receptor Activation

The pregnane X receptor (PXR) is a master regulator of xenobiotic clearance and is implicated in deleterious drug interactions (e.g., acetaminophen hepatotoxicity) and cancer drug resistance. However, small-molecule targeting of this receptor has been difficult; to date, directed synthesis of a rela...

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Autors principals: Venkatesh, Madhukumar, Wang, Hongwei, Cayer, Julie, Leroux, Melissa, Salvail, Dany, Das, Bhaskar, Wrobel, Jay E., Mani, Sridhar
Format: Artigo
Idioma:Inglês
Publicat: The American Society for Pharmacology and Experimental Therapeutics 2011
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Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC3127530/
https://ncbi.nlm.nih.gov/pubmed/21464197
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1124/mol.111.071787
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