Загрузка...

Evaluation of NTF1836 as an inhibitor of the mycothiol biosynthetic enzyme MshC in growing and non-replicating Mycobacterium tuberculosis

The mycothiol biosynthesis enzyme MshC catalyzes the ligation of cysteine with the pseudodisaccharide GlcN-Ins and has been identified as an essential enzyme in Mycobacterium tuberculosis. We now report on the development of NTF1836 as a micromolar inhibitor of MshC. Using commercial libaries, we co...

Полное описание

Сохранить в:
Библиографические подробности
Главные авторы: Newton, Gerald L., Buchmeier, Nancy, La Clair, James J., Fahey, Robert C.
Формат: Artigo
Язык:Inglês
Опубликовано: 2011
Предметы:
Online-ссылка:https://ncbi.nlm.nih.gov/pmc/articles/PMC3123436/
https://ncbi.nlm.nih.gov/pubmed/21665483
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.bmc.2011.05.028
Метки: Добавить метку
Нет меток, Требуется 1-ая метка записи!