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Dasatinib enhances megakaryocyte differentiation but inhibits platelet formation

Dasatinib is a novel, potent, ATP-competitive inhibitor of Bcr-Abl, cKIT, and Src family kinases that exhibits efficacy in patients with imatinib-resistant chronic myelogenous leukemia. Dasatinib treatment is associated with mild thrombocytopenia and an increased risk of bleeding, but its biological...

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Bibliografiske detaljer
Main Authors: Mazharian, Alexandra, Ghevaert, Cedric, Zhang, Lin, Massberg, Steffen, Watson, Steve P.
Format: Artigo
Sprog:Inglês
Udgivet: American Society of Hematology 2011
Fag:
Online adgang:https://ncbi.nlm.nih.gov/pmc/articles/PMC3109542/
https://ncbi.nlm.nih.gov/pubmed/21385851
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1182/blood-2010-12-326850
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