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Improved Total Synthesis of the Potent HDAC Inhibitor FK228 (FR-901228)

[Image: see text] A scaleable synthesis of the potent histone deacetylase (HDAC) inhibitor FK228 is described. A reliable strategy for preparing the key β-hydroxy mercapto heptenoic acid partner was accomplished in nine steps and 13% overall yield. A Noyori asymmetric hydrogen-transfer reaction esta...

Ausführliche Beschreibung

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Bibliographische Detailangaben
Hauptverfasser: Greshock, Thomas J., Johns, Deidre M., Noguchi, Yasuo, Williams, Robert M.
Format: Artigo
Sprache:Inglês
Veröffentlicht: 2008
Schlagworte:
Online Zugang:https://ncbi.nlm.nih.gov/pmc/articles/PMC3097137/
https://ncbi.nlm.nih.gov/pubmed/18205373
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/ol702957z
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