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GS-8374, a Novel HIV Protease Inhibitor, Does Not Alter Glucose Homeostasis in Cultured Adipocytes or in a Healthy-Rodent Model System

Adverse effects induced by HIV protease inhibitors (PIs) are a significant factor in limiting their clinical success. PIs directly contribute to peripheral insulin resistance and alterations in lipid metabolism. GS-8374 is a novel PI with potent antiretroviral activity and a favorable resistance pro...

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Détails bibliographiques
Auteurs principaux: Hruz, Paul W., Yan, Qingyun, Tsai, Luong, Koster, Joseph, Xu, Lianhong, Cihlar, Tomas, Callebaut, Christian
Format: Artigo
Langue:Inglês
Publié: American Society for Microbiology (ASM) 2011
Sujets:
Accès en ligne:https://ncbi.nlm.nih.gov/pmc/articles/PMC3067185/
https://ncbi.nlm.nih.gov/pubmed/21245443
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1128/AAC.01184-10
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