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Synthesis and Biological Evaluation of Apogossypolone Derivatives as Pan-active Inhibitors of Anti-apoptotic B-Cell Lymphoma/Leukemia-2 (Bcl-2) Family Proteins

Overexpression of anti-apoptotic Bcl-2 family proteins is commonly related with tumor maintenance, progression, and chemoresistance. Inhibition of these anti-apoptotic proteins is an attractive approach for cancer therapy. Guided by nuclear magnetic resonance (NMR) binding assays, a series of 5, 5′...

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Détails bibliographiques
Auteurs principaux: Wei, Jun, Kitada, Shinichi, Stebbins, John L., Placzek, William, Zhai, Dayong, Wu, Bainan, Rega, Michele F., Zhang, Ziming, Cellitti, Jason, Yang, Li, Dahl, Russell, Reed, John C., Pellecchia, Maurizio
Format: Artigo
Langue:Inglês
Publié: 2010
Sujets:
Accès en ligne:https://ncbi.nlm.nih.gov/pmc/articles/PMC3059195/
https://ncbi.nlm.nih.gov/pubmed/21033669
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/jm100746q
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