Llwytho...

Potent and Selective Photo-inactivation of Proteins With Peptoid-Ruthenium Conjugates

Advances in high-throughput screening now enable the rapid discovery of bioactive small molecules, but these primary hits almost always exhibit modest potency. We report a strategy for the transformation of these hits into much more potent inhibitors without compound optimization. Appending a deriva...

Disgrifiad llawn

Wedi'i Gadw mewn:
Manylion Llyfryddiaeth
Prif Awduron: Lee, Jiyong, Udugamasooriya, D. Gomika, Lim, Hyun-Suk, Kodadek, Thomas
Fformat: Artigo
Iaith:Inglês
Cyhoeddwyd: 2010
Pynciau:
Mynediad Ar-lein:https://ncbi.nlm.nih.gov/pmc/articles/PMC3049443/
https://ncbi.nlm.nih.gov/pubmed/20228793
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1038/nchembio.333
Tagiau: Ychwanegu Tag
Dim Tagiau, Byddwch y cyntaf i dagio'r cofnod hwn!