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Copper-free click conjugation of methotrexate to a PAMAM dendrimer platform

The synthesis of a generation 5 (G5) poly(amidoamine) (PAMAM) dendrimer platform having cyclooctyne ligands that were subsequently be used for a copper-free Huisgen 1,3-dipolar cycloaddition (click reaction) with azido modified methotrexate is described. The G5 PAMAM dendrimer was first partially (7...

Ausführliche Beschreibung

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Bibliographische Detailangaben
Hauptverfasser: Huang, Baohua, Desai, Ankur, Zong, Hong, Tang, Shengzhuang, Leroueil, Pascale, Baker, James R.
Format: Artigo
Sprache:Inglês
Veröffentlicht: 2011
Schlagworte:
Online Zugang:https://ncbi.nlm.nih.gov/pmc/articles/PMC3048335/
https://ncbi.nlm.nih.gov/pubmed/21383864
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.tetlet.2010.12.025
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