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Design and Synthesis of Potent HIV-1 Protease Inhibitors Incorporating Hexahydrofuropyranol-derived High Affinity P(2) ligands: Structure-activity Studies and Biological Evaluation

The design, synthesis, and evaluation of a new series of hexahydrofuropyran-derived HIV-1 protease inhibitors are described. We have designed a stereochemically defined hexahydrofuropyranol-derived urethane as the P2-ligand. The current ligand is designed based upon the X-ray structure of 1a-bound H...

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Hlavní autoři: Ghosh, Arun K., Chapsal, Bruno D., Baldridge, Abigail, Steffey, Melinda P., Walters, D. Eric, Koh, Yasuhiro, Amano, Masayuki, Mitsuya, Hiroaki
Médium: Artigo
Jazyk:Inglês
Vydáno: 2010
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On-line přístup:https://ncbi.nlm.nih.gov/pmc/articles/PMC3024462/
https://ncbi.nlm.nih.gov/pubmed/21194227
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/jm1012787
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