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Structure-Based Design, Synthesis and Structure-Activity Relationship Studies of HIV-1 Protease Inhibitors Incorporating Phenyloxazolidinones

A series of new HIV-1 protease inhibitors with the hydroxyethylamine core and different phenyloxazolidinone P2 ligands were designed and synthesized. Variation of phenyl substitutions at the P2 and P2′ moieties significantly affected the inhibitors’ binding affinity and antiviral potency. In general...

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Detalhes bibliográficos
Main Authors: Ali, Akbar, Kiran Kumar Reddy, G. S., Nalam, Madhavi N. L., Anjum, Saima Ghafoor, Cao, Hong, Schiffer, Celia A., Rana, Tariq M.
Formato: Artigo
Idioma:Inglês
Publicado em: 2010
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC2996262/
https://ncbi.nlm.nih.gov/pubmed/20958050
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/jm1008743
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