A carregar...

Rational Design and Simple Chemistry Yield a Superior, Neuroprotective HDAC6 Inhibitor, Tubastatin A

Structure-based drug design combined with homology modeling techniques were used to develop potent inhibitors of HDAC6 that display superior selectivity for the HDAC6 isozyme compared to other inhibitors. These inhibitors can be assembled in a few synthetic steps, as thus are readily scaled up for i...

ver descrição completa

Na minha lista:
Detalhes bibliográficos
Main Authors: Butler, Kyle V, Kalin, Jay, Brochier, Camille, Vistoli, Guilio, Langley, Brett, Kozikowski, Alan P
Formato: Artigo
Idioma:Inglês
Publicado em: 2010
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC2916045/
https://ncbi.nlm.nih.gov/pubmed/20614936
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/ja102758v
Tags: Adicionar Tag
Sem tags, seja o primeiro a adicionar uma tag!