Wird geladen...

Using Ligand-Based Virtual Screening to Allosterically Stabilize the Activated State of a GPCR

G-protein coupled receptors (GPCRs) play an essential role in many biological processes. Despite an increase in the number of solved X-ray crystal structures of GPCRs, capturing a GPCR in its activated state for structural analysis has proven to be difficult. An unexplored paradigm is stabilization...

Ausführliche Beschreibung

Gespeichert in:
Bibliographische Detailangaben
Hauptverfasser: Taylor, Christina M., Rockweiler, Nicole B., Liu, Cassie, Rikimaru, Loryn, Tunemalm, Anna-Karin, Kisselev, Oleg G., Marshall, Garland R.
Format: Artigo
Sprache:Inglês
Veröffentlicht: 2010
Schlagworte:
Online Zugang:https://ncbi.nlm.nih.gov/pmc/articles/PMC2911999/
https://ncbi.nlm.nih.gov/pubmed/20659113
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1111/j.1747-0285.2009.00944.x
Tags: Tag hinzufügen
Keine Tags, Fügen Sie den ersten Tag hinzu!