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Macrocyclic Pyridyl Polyoxazoles: Selective RNA and DNA G-Quadruplex Ligands as Antitumor Agents

The synthesis of a series of 24-membered pyridine-containing polyoxazole macrocycles is described. Seventeen new macrocycles were evaluated for cytotoxic activity against RPMI 8402, KB-3, and KB-3 cell lines that overexpress the efflux transporters MDR1 (KBV-1) and BCRP (KBH5.0). Macrocycles in whic...

Täydet tiedot

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Bibliografiset tiedot
Päätekijät: Rzuczek, Suzanne G., Pilch, Daniel S., Liu, Angela, Liu, Leroy, LaVoie, Edmond J., Rice, Joseph E.
Aineistotyyppi: Artigo
Kieli:Inglês
Julkaistu: 2010
Aiheet:
Linkit:https://ncbi.nlm.nih.gov/pmc/articles/PMC2865558/
https://ncbi.nlm.nih.gov/pubmed/20359224
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/jm1000612
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