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Chk1 C-terminal regulatory phosphorylation mediates checkpoint activation via derepression of Chk1 catalytic activity

Chk1 is phosphorylated within its C-terminal regulatory domain by the upstream ATM/ ATR kinases during checkpoint activation, however how this modulates Chk1 function is poorly understood. Here, we show that Chk1 kinase activity is rapidly stimulated in a cell cycle phase-specific manner in response...

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Autori principali: Walker, M, Black, EJ, Oehler, V, Gillespie, DA, Scott, MT
Natura: Artigo
Lingua:Inglês
Pubblicazione: 2009
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC2857325/
https://ncbi.nlm.nih.gov/pubmed/19421147
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1038/onc.2009.102
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