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Rational design of dualsteric GPCR ligands: quests and promise

Dualsteric ligands represent a novel mode of targeting G protein-coupled receptors (GPCRs). These compounds attach simultaneously to both, the orthosteric transmitter binding site and an additional allosteric binding area of a receptor protein. This approach allows the exploitation of favourable cha...

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Dettagli Bibliografici
Autori principali: Mohr, Klaus, Tränkle, Christian, Kostenis, Evi, Barocelli, Elisabetta, De Amici, Marco, Holzgrabe, Ulrike
Natura: Artigo
Lingua:Inglês
Pubblicazione: Blackwell Publishing Ltd 2010
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC2839259/
https://ncbi.nlm.nih.gov/pubmed/20136835
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1111/j.1476-5381.2009.00601.x
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