Wird geladen...

Rational design of dualsteric GPCR ligands: quests and promise

Dualsteric ligands represent a novel mode of targeting G protein-coupled receptors (GPCRs). These compounds attach simultaneously to both, the orthosteric transmitter binding site and an additional allosteric binding area of a receptor protein. This approach allows the exploitation of favourable cha...

Ausführliche Beschreibung

Gespeichert in:
Bibliographische Detailangaben
Hauptverfasser: Mohr, Klaus, Tränkle, Christian, Kostenis, Evi, Barocelli, Elisabetta, De Amici, Marco, Holzgrabe, Ulrike
Format: Artigo
Sprache:Inglês
Veröffentlicht: Blackwell Publishing Ltd 2010
Schlagworte:
Online Zugang:https://ncbi.nlm.nih.gov/pmc/articles/PMC2839259/
https://ncbi.nlm.nih.gov/pubmed/20136835
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1111/j.1476-5381.2009.00601.x
Tags: Tag hinzufügen
Keine Tags, Fügen Sie den ersten Tag hinzu!