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Screening-based discovery of drug-like O-GlcNAcase inhibitor scaffolds

O-GlcNAcylation is an essential posttranslational modification in metazoa. Modulation of O-GlcNAc levels with small molecule inhibitors of O-GlcNAc hydrolase (OGA) is a useful strategy to probe the role of this modification in a range of cellular processes. Here we report the discovery of novel, low...

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Main Authors: Dorfmueller, Helge C., van Aalten, Daan M.F.
格式: Artigo
語言:Inglês
出版: Elsevier Science B.V 2010
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在線閱讀:https://ncbi.nlm.nih.gov/pmc/articles/PMC2828546/
https://ncbi.nlm.nih.gov/pubmed/20026047
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.febslet.2009.12.020
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