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Roscovitine Binds to Novel L-channel (Ca(V)1.2) Sites That Separately Affect Activation and Inactivation

L-type (Ca(V)1.2) calcium channel antagonists play an important role in the treatment of cardiovascular disease. (R)-Roscovitine, a trisubstituted purine, has been shown to inhibit L-currents by slowing activation and enhancing inactivation. This study utilized molecular and pharmacological approach...

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Detalhes bibliográficos
Main Authors: Yarotskyy, Viktor, Gao, Guofeng, Du, Lei, Ganapathi, Sindura B., Peterson, Blaise Z., Elmslie, Keith S.
Formato: Artigo
Idioma:Inglês
Publicado em: American Society for Biochemistry and Molecular Biology 2010
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC2804190/
https://ncbi.nlm.nih.gov/pubmed/19887376
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1074/jbc.M109.076448
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