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Roscovitine, a cyclin-dependent kinase inhibitor, affects several gating mechanisms to inhibit cardiac L-type (Ca((V))1.2) calcium channels

BACKGROUND AND PURPOSE: L-type calcium channels (Ca ((V))1.2) play an important role in cardiac contraction. Roscovitine, a cyclin-dependent kinase inhibitor and promising anticancer drug, has been shown to affect Ca ((V))1.2 by inhibiting current amplitude and slowing activation. This research inve...

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Bibliografski detalji
Glavni autori: Yarotskyy, V, Elmslie, K S
Format: Artigo
Jezik:Inglês
Izdano: Nature Publishing Group 2007
Teme:
Online pristup:https://ncbi.nlm.nih.gov/pmc/articles/PMC2042960/
https://ncbi.nlm.nih.gov/pubmed/17700718
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1038/sj.bjp.0707414
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