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X-ray Crystallographic Analysis of α-Ketoheterocycle Inhibitors Bound to a Humanized Variant of Fatty Acid Amide Hydrolase

Three cocrystal X-ray structures of the α-ketoheterocycle inhibitors 3–5 bound to a humanized variant of fatty acid amide hydrolase (FAAH) are disclosed and comparatively discussed alongside those of 1 (OL-135) and its isomer 2. These five X-ray structures systematically probe each of the three acti...

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Detalhes bibliográficos
Main Authors: Mileni, Mauro, Garfunkle, Joie, Ezzili, Cyrine, Kimball, F. Scott, Cravatt, Benjamin F., Stevens, Raymond C., Boger, Dale L.
Formato: Artigo
Idioma:Inglês
Publicado em: 2010
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC2804032/
https://ncbi.nlm.nih.gov/pubmed/19924997
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/jm9012196
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