Učitavanje...

Exploration of a fundamental substituent effect of α-ketoheterocycle enzyme inhibitors: potent and selective inhibitors of fatty acid amide hydrolase

A series of C4 substituted α-ketooxazoles were examined as inhibitors of the serine hydrolase fatty acid amide hydrolase in efforts that further define and generalize a fundamental substituent effect on enzyme inhibitory potency. Thus, a plot of the Hammett σ(m) versus –log K(i) provided a linear co...

Cijeli opis

Spremljeno u:
Bibliografski detalji
Glavni autori: DeMartino, Jessica K., Garfunkle, Joie, Hochstatter, Dustin G., Cravatt, Benjamin F., Boger, Dale L.
Format: Artigo
Jezik:Inglês
Izdano: 2008
Teme:
Online pristup:https://ncbi.nlm.nih.gov/pmc/articles/PMC2582052/
https://ncbi.nlm.nih.gov/pubmed/18639454
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.bmcl.2008.06.084
Oznake: Dodaj oznaku
Bez oznaka, Budi prvi tko označuje ovaj zapis!