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Novel Molecular Determinants in the Pore Region of Sodium Channels Regulate Local Anesthetic Binding

The pore of the Na(+) channel is lined by asymmetric loops formed by the linkers between the fifth and sixth transmembrane segments (S5-S6). We investigated the role of the N-terminal portion (SS1) of the S5-S6 linkers in channel gating and local anesthetic (LA) block using site-directed cysteine mu...

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Autors principals: Yamagishi, Toshio, Xiong, Wei, Kondratiev, Andre, Vélez, Patricio, Méndez-Fitzwilliam, Ailsa, Balser, Jeffrey R., Marbán, Eduardo, Tomaselli, Gordon F.
Format: Artigo
Idioma:Inglês
Publicat: The American Society for Pharmacology and Experimental Therapeutics 2009
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Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC2769053/
https://ncbi.nlm.nih.gov/pubmed/19620257
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1124/mol.109.055863
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