Conformationally constrained opioid ligands: The Dmt-Aba and Dmt-Aia vs. Dmt-Tic scaffold

Replacement of the constrained phenylalanine analogue 1,2,3,4-tetrahydroisoquinoline-3-carboxylic acid (Tic) in the opioid Dmt-Tic-Gly-NH-Bn scaffold by the 4-amino-1,2,4,5-tetrahydro-indolo[2,3-c]azepin-3-one (Aia) and 4-amino-1,2,4,5-tetrahydro-2-benzazepin-3-one (Aba) scaffolds has led to the dis...

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Bibliografische gegevens
Hoofdauteurs: Ballet, Steven, Feytens, Debby, De Wachter, Rien, De Vlaeminck, Magali, Marczak, Ewa D., Salvadori, Severo, de Graaf, Chris, Rognan, Didier, Negri, Lucia, Lattanzi, Roberta, Lazarus, Lawrence H., Tourwé, Dirk, Balboni, Gianfranco
Formaat: Artigo
Taal:Inglês
Gepubliceerd in: 2008
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Article
Online toegang:https://ncbi.nlm.nih.gov/pmc/articles/PMC2742322/
https://ncbi.nlm.nih.gov/pubmed/19062273
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.bmcl.2008.11.051
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