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Agonist-induced internalization and downregulation of gonadotropin-releasing hormone receptors
Gonadotropin-releasing hormone (GnRH) acts via seven transmembrane receptors to stimulate gonadotropin secretion. Sustained stimulation desensitizes GnRH receptor (GnRHR)-mediated gonadotropin secretion, and this underlies agonist use in hormone-dependent cancers. Since type I mammalian GnRHR do not...
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| Autors principals: | , , , |
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| Format: | Artigo |
| Idioma: | Inglês |
| Publicat: |
American Physiological Society
2009
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| Matèries: | |
| Accés en línia: | https://ncbi.nlm.nih.gov/pmc/articles/PMC2740399/ https://ncbi.nlm.nih.gov/pubmed/19587220 https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1152/ajpcell.00166.2009 |
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