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Differential Regulation of Receptor Activation and Agonist Selectivity by Highly Conserved Tryptophans in the Nicotinic Acetylcholine Receptor Binding Site

We have shown previously that a highly conserved Tyr in the nicotinic acetylcholine receptor (nAChR) ligand-binding domain (LBD) (α7 Tyr188 or α4 Tyr195) differentially regulates the activity of acetylcholine (ACh) and the α7-selective agonist 3-(4-hydroxy,2-methoxybenzylidene)anabaseine (4OH-GTS-21...

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Библиографические подробности
Главные авторы: Williams, Dustin K., Stokes, Clare, Horenstein, Nicole A., Papke, Roger L.
Формат: Artigo
Язык:Inglês
Опубликовано: American Society for Pharmacology and Experimental Therapeutics 2009
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Online-ссылка:https://ncbi.nlm.nih.gov/pmc/articles/PMC2700159/
https://ncbi.nlm.nih.gov/pubmed/19339660
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1124/jpet.109.151225
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