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A Cremophor-Free Formulation for Tanespimycin (17-AAG) using PEO-b-PDLLA Micelles: Characterization and Pharmacokinetics in Rats

Tanespimycin (17-allylamino-17-demethoxygeldanamycin or 17-AAG) is a promising heat shock protein 90 inhibitor currently undergoing clinical trials for the treatment of cancer. Despite its selective mechanism of action on cancer cells, 17-AAG faces challenging issues due to its poor aqueous solubili...

Deskribapen osoa

Gorde:
Xehetasun bibliografikoak
Egile Nagusiak: Xiong, May P., Yáñez, Jaime A., Kwon, Glen S., Davies, Neal M., Forrest, M. Laird
Formatua: Artigo
Hizkuntza:Inglês
Argitaratua: 2009
Gaiak:
Sarrera elektronikoa:https://ncbi.nlm.nih.gov/pmc/articles/PMC2649998/
https://ncbi.nlm.nih.gov/pubmed/18752263
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1002/jps.21509
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