Synthesis of 3,6-bis[H-Tyr/H-Dmt-NH(CH(2))(m,n)]-2(1H)pyrazinone derivatives: function of alkyl chain length on opioid activity

Lignende værker

• Design and Synthesis of Opioidmimetics Containing 2′,6′-Dimethyl-l-tyrosine and a Pyrazinone-Ring Platform
  af: Shiotani, Kimitaka, et al.
  Udgivet: (2007)
• Conversion of the Potent δ-Opioid Agonist H-Dmt-Tic-NH-CH(2)-Bid into δ-Opioid Antagonists by N(1)-Benzimidazole Alkylation1
  af: Balboni, Gianfranco, et al.
  Udgivet: (2005)
• Bifunctional [2’,6’-Dimethyl-l-tyrosine(1)]Endomorphin-2 Analogues Substituted at Position 3 with Alkylated Phenylalanine Derivatives Yield Potent Mixed μ-Agonist/δ-Antagonist and Dual μ-/δ-Agonist Opioid Ligands
  af: Li, Tingyou, et al.
  Udgivet: (2007)
• Role of Benzimidazole (Bid) in the δ Opioid Agonist Pseudopeptide H-Dmt-Tic-NH-CH(2)-Bid (UFP-502)
  af: Salvadori, Severo, et al.
  Udgivet: (2007)
• Inhibition of the Development of Morphine Tolerance by a Potent Dual μ-/δ-Opioid Antagonist, H-Dmt-Tic-Lys-NH-CH(2)-Ph
  af: Jinsmaa, Yunden, et al.
  Udgivet: (2008)