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Variety of Antiprion Compounds Discovered through an In Silico Screen Based on Cellular-Form Prion Protein Structure: Correlation between Antiprion Activity and Binding Affinity

Transmissible spongiform encephalopathies are associated with the conformational conversion of the prion protein from the cellular form (PrP(C)) to the scrapie form. This process could be disrupted by stabilizing the PrP(C) conformation, using a specific ligand identified as a chemical chaperone. To...

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Gorde:
Xehetasun bibliografikoak
Egile Nagusiak: Hosokawa-Muto, Junji, Kamatari, Yuji O., Nakamura, Hironori K., Kuwata, Kazuo
Formatua: Artigo
Hizkuntza:Inglês
Argitaratua: American Society for Microbiology (ASM) 2009
Gaiak:
Sarrera elektronikoa:https://ncbi.nlm.nih.gov/pmc/articles/PMC2630596/
https://ncbi.nlm.nih.gov/pubmed/19015328
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1128/AAC.01112-08
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