Chargement en cours...

Mechanism-based inhibitors of MenE, an acyl-CoA synthetase involved in bacterial menaquinone biosynthesis

Menaquinone (vitamin K(2)) is an essential component of the electron transfer chain in many pathogens, including Mycobacterium tuberculosis and Staphylococcus aureus, and menaquinone biosynthesis is a potential target for antibiotic drug discovery. We report herein a series of mechanism-based inhibi...

Description complète

Enregistré dans:
Détails bibliographiques
Auteurs principaux: Lu, Xuequan, Zhang, Huaning, Tonge, Peter J., Tan, Derek S.
Format: Artigo
Langue:Inglês
Publié: 2008
Sujets:
Accès en ligne:https://ncbi.nlm.nih.gov/pmc/articles/PMC2628629/
https://ncbi.nlm.nih.gov/pubmed/18762421
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.bmcl.2008.07.130
Tags: Ajouter un tag
Pas de tags, Soyez le premier à ajouter un tag!