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Stoichiometry and Physical Chemistry of Promiscuous Aggregate-Based Inhibitors

Many false positives in early drug discovery owe to nonspecific inhibition by colloid-like aggregates of organic molecules. Despite their prevalence, little is known about aggregate concentration, structure, or dynamic equilibrium; the binding mechanism, stoichiometry with, and affinity for enzymes...

Ausführliche Beschreibung

Gespeichert in:
Bibliographische Detailangaben
Hauptverfasser: Coan, Kristin E. D., Shoichet, Brian K.
Format: Artigo
Sprache:Inglês
Veröffentlicht: 2008
Schlagworte:
Online Zugang:https://ncbi.nlm.nih.gov/pmc/articles/PMC2627561/
https://ncbi.nlm.nih.gov/pubmed/18588298
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/ja802977h
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