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Human P2Y(6) Receptor: Molecular Modeling Leads to the Rational Design of a Novel Agonist Based on a Unique Conformational Preference

Combining molecular dynamics (MD) in a hydrated phospholipids (DOPC) bilayer, Monte Carlo search, and synthesis of locked nucleotide analogues we discovered that the Southern conformation of the ribose is preferred for ligand recognition by the P2Y(6) receptor. 2′-Deoxy-(S)-methanocarbaUDP was found...

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Autors principals: Costanzi, Stefano, Joshi, Bhalchandra V., Maddileti, Savitri, Mamedova, Liaman, Gonzalez-Moa, Maria J., Marquez, Victor E., Harden, T. Kendall, Jacobson, Kenneth A.
Format: Artigo
Idioma:Inglês
Publicat: 2005
Matèries:
Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC2583457/
https://ncbi.nlm.nih.gov/pubmed/16366591
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/jm050911p
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