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Allosteric Modulation of the Dopamine Receptor by Conformationally Constrained Type VI β-Turn Peptidomimetics of Pro-Leu-Gly-NH(2)

A peptidomimetic of Pro-Leu-Pro-NH(2), 7, possessing an indolizidinone type VI β-turn mimic was synthesized via improved high-yielding protocols for the preparation and Cbz-protection of α-allyl proline. Bicyclic peptidomimetic 7 and spirobicylic peptidomimetic 8 enhanced the binding of [(3)H]N-prop...

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Détails bibliographiques
Auteurs principaux: Vartak, Ashish, Skoblenick, Kevin, Thomas, Nancy, Mishra, Ram K., Johnson, Rodney L.
Format: Artigo
Langue:Inglês
Publié: 2007
Sujets:
Accès en ligne:https://ncbi.nlm.nih.gov/pmc/articles/PMC2529021/
https://ncbi.nlm.nih.gov/pubmed/18052024
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/jm070895r
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