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A unique class of duocarmycin and CC-1065 analogues subject to reductive activation

N-Acyl O-amino phenol derivatives of CBI-TMI and CBI-indole(2) are reported as prototypical members of a new class of reductively activated prodrugs of the duocarmycin and CC-1065 class of antitumor agents. The expectation being that hypoxic tumor environments, with their higher reducing capacity, c...

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Bibliografische gegevens
Hoofdauteurs: Jin, Wei, Trzupek, John D., Rayl, Thomas J., Broward, Melinda A., Vielhauer, George A., Weir, Scott J., Hwang, Inkyu, Boger, Dale L.
Formaat: Artigo
Taal:Inglês
Gepubliceerd in: 2007
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Online toegang:https://ncbi.nlm.nih.gov/pmc/articles/PMC2519901/
https://ncbi.nlm.nih.gov/pubmed/18020335
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/ja075398e
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