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Design, Synthesis, and Evaluation of Duocarmycin O-Amino Phenol Prodrugs Subject to Tunable Reductive Activation

A series of N-acyl O-amino derivatives of seco-CBI-indole(2) are reported and examined as prototypical members of a unique class of reductively activated (cleaved) prodrugs of the duocarmycin and CC-1065 family of antitumor agents. These prodrugs were designed to be potentially preferentially activa...

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Main Authors: Lajiness, James P., Robertson, William M., Dunwiddie, Irene, Broward, Melinda A., Vielhauer, George A., Weir, Scott J., Boger, Dale L.
Formato: Artigo
Idioma:Inglês
Publicado: 2010
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Acceso en liña:https://ncbi.nlm.nih.gov/pmc/articles/PMC2974002/
https://ncbi.nlm.nih.gov/pubmed/20942408
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/jm1010397
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