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Gossypol, a BH3 mimetic, induces apoptosis in chronic lymphocytic leukemia cells

Gossypol, a cottonseed extract derivative, acts as a BH3-mimetic, binding to the BH3 pocket of antiapoptotic proteins and displacing pro-death partners to induce apoptosis. However, knowledge on the molecular underpinnings of its downstream effects is limited. Since chronic lymphocytic leukemia (CLL...

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Hlavní autoři: Balakrishnan, Kumudha, Wierda, William G., Keating, Michael J., Gandhi, Varsha
Médium: Artigo
Jazyk:Inglês
Vydáno: American Society of Hematology 2008
Témata:
On-line přístup:https://ncbi.nlm.nih.gov/pmc/articles/PMC2518898/
https://ncbi.nlm.nih.gov/pubmed/18566329
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1182/blood-2007-12-126946
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