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Kinetics and Mechanisms of Activation of α-Amino Acid Ester Prodrugs of Camptothecins

The α-amino acid ester prodrugs of the antitumor agent camptothecin and a more potent, lipophilic silatecan analog, DB-67, have been shown by NMR spectroscopy and quantitative kinetic analyses to undergo quantitative conversion to their pharmacologically active lactones via a non-enzymatic mechanism...

Ausführliche Beschreibung

Gespeichert in:
Bibliographische Detailangaben
Hauptverfasser: Song, Lin, Bevins, Robert, Anderson, Bradley D.
Format: Artigo
Sprache:Inglês
Veröffentlicht: 2006
Schlagworte:
Online Zugang:https://ncbi.nlm.nih.gov/pmc/articles/PMC2516925/
https://ncbi.nlm.nih.gov/pubmed/16821794
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/jm060016l
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