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How ATP Inhibits the Open K(ATP) Channel

ATP-sensitive potassium (K(ATP)) channels are composed of four pore-forming Kir6.2 subunits and four regulatory SUR1 subunits. Binding of ATP to Kir6.2 leads to inhibition of channel activity. Because there are four subunits and thus four ATP-binding sites, four binding events are possible. ATP bind...

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Autori principali: Craig, Tim J., Ashcroft, Frances M., Proks, Peter
Natura: Artigo
Lingua:Inglês
Pubblicazione: The Rockefeller University Press 2008
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC2442177/
https://ncbi.nlm.nih.gov/pubmed/18591420
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1085/jgp.200709874
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