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In vitro evaluation of amino acid prodrugs of novel antitumour 2-(4-amino-3-methylphenyl)benzothiazoles

Novel 2-(4-aminophenyl)benzothiazoles possess highly selective, potent antitumour properties in vitro and in vivo. They induce and are biotransformed by cytochrome P450 (CYP) 1A1 to putative active as well as inactive metabolites. Metabolic inactivation of the molecule has been thwarted by isosteric...

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Détails bibliographiques
Auteurs principaux: Bradshaw, T D, Chua, M-S, Browne, H L, Trapani, V, Sausville, E A, Stevens, M F G
Format: Artigo
Langue:Inglês
Publié: Nature Publishing Group 2002
Sujets:
Accès en ligne:https://ncbi.nlm.nih.gov/pmc/articles/PMC2375326/
https://ncbi.nlm.nih.gov/pubmed/11953897
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1038/sj.bjc.6600225
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